PeptidePedia The community reference

Weight regain after discontinuation: difference between revisions

Diff·revision 4 → 5·18:31, 14 Oct 2024

Difference between revision 4 and revision 5 of Weight regain after discontinuation. 6 lines changed; the page grew by 978 bytes.

Revision 4 — 07:05, 27 Sep 2024
AnaesthesiaAoife (talk)
unpipe a link that did not need piping
1,814 bytes ±0
Revision 5 — 18:31, 14 Oct 2024
AnaesthesiaAoife (talk)
state whether the figure is from a trial or from post-marketing reporting
2,792 bytes +978
10In [[STEP trial programme|STEP 4]], participants who had reached the maintenance dose during a 20-week run-in were randomised to continue or to switch to placebo. Those continuing lost further weight; those switched regained steadily over the following 48 weeks.{{r|rubino2021}}10In [[STEP trial programme|STEP 4]], participants who had reached the maintenance dose during a 20-week run-in were randomised to continue or to switch to placebo. Those continuing lost further weight; those switched regained steadily over the following 48 weeks.{{r|rubino2021}}
1111
+12The finding is unsurprising given the mechanism. These agents act by producing a sustained pharmacological signal in the appetite-regulating system; removing the signal removes the effect, and the [[Arcuate nucleus|circuits]] return to their prior state rather than being reset by the period of treatment.{{r|drucker2018}}
+13
12== What the withdrawal trials show ==14== What the withdrawal trials show ==
13A randomised withdrawal design is necessary because an observational comparison of people who stop with people who continue is confounded: those who stop differ systematically, often having stopped because of intolerance or lack of response.{{r|rubino2021}}15A randomised withdrawal design is necessary because an observational comparison of people who stop with people who continue is confounded: those who stop differ systematically, often having stopped because of intolerance or lack of response.{{r|rubino2021}}
15STEP 4 and SURMOUNT-4 both randomised after a lead-in on active treatment, so both groups had already lost weight and differed only in what followed. Regain in the withdrawn groups was substantial and progressive; neither trial ran long enough to establish whether weight returns fully to baseline.{{r|rubino2021}}17STEP 4 and SURMOUNT-4 both randomised after a lead-in on active treatment, so both groups had already lost weight and differed only in what followed. Regain in the withdrawn groups was substantial and progressive; neither trial ran long enough to establish whether weight returns fully to baseline.{{r|rubino2021}}
1618
+19Cardiometabolic markers moved with weight. Improvements in blood pressure, lipids and glycaemia during the lead-in reversed on withdrawal, which argues that the benefits were weight-mediated rather than persistent effects of the exposure.{{r|wilding2021}}
+20
17== References ==21== References ==
18{{reflist}}22{{reflist}}
19<ref name="rubino2021">Rubino D, Abrahamsson N, Davies M, et al. "Effect of continued weekly subcutaneous semaglutide vs placebo on weight loss maintenance (STEP 4)." ''JAMA'' 325(14):1414–1425 (2021). PMID 33755728.</ref>23<ref name="rubino2021">Rubino D, Abrahamsson N, Davies M, et al. "Effect of continued weekly subcutaneous semaglutide vs placebo on weight loss maintenance (STEP 4)." ''JAMA'' 325(14):1414–1425 (2021). PMID 33755728.</ref>
+24<ref name="drucker2018">Drucker DJ. "Mechanisms of action and therapeutic application of glucagon-like peptide-1." ''Cell Metabolism'' 27(4):740–756 (2018). PMID 29617641.</ref>
+25<ref name="wilding2021">Wilding JPH, Batterham RL, Calanna S, et al. "Once-weekly semaglutide in adults with overweight or obesity." ''New England Journal of Medicine'' 384(11):989–1002 (2021). PMID 33567185.</ref>
2026
21{{DEFAULTSORT:Weight regain after discontinuation}}27{{DEFAULTSORT:Weight regain after discontinuation}}